Tag

Photopharmacology

All articles tagged with #photopharmacology

science2 hours ago

Light-Activated Drugs Restore Sight in Blind Mice Without Implants

Researchers developed photoswitchable small-molecule drugs (prosthe6) that mimic photoreceptor signaling and reactivate intact retinal circuits in blind mice and zebrafish. Delivered by eye injections or eye drops, these compounds restore light responses under normal indoor lighting without implants or genetic modification, effectively reviving basic visual behavior in animal models; two compounds, prosthe6-12 and prosthe6-15, showed especially strong results. Human testing has not begun; safety and formulation work continues with the goal of a noninvasive, drug-based vision restoration approach applicable to many retinal diseases.

Light-Activated PROTACs Wake Dormant Lung Cancer Cells
science1 month ago

Light-Activated PROTACs Wake Dormant Lung Cancer Cells

Researchers engineered light-switchable PROTACs that degrade the glucocorticoid receptor, which can drive cancer cells into a dormancy state. In lab tests with human lung cancer cells, the active E-form of two lead compounds destroyed the receptor and reversed dormancy-linked gene activity, while the inactive Z-form largely did nothing. The switch is controlled by different wavelengths of light, though UV light was used in experiments to keep the inactive form stable; these wavelengths do not penetrate tissue well, posing a major barrier to clinical use. The work is early-stage and lab-only, with future goals to develop red/near-infrared–sensitive versions for deeper tissue targeting and eventual therapeutic applications.